• Article  

      Ciprofloxacin conjugated to diphenyltin(iv): a novel formulation with enhanced antimicrobial activity 

      Chrysouli, M. P.; Banti, Christina N.; Kourkoumelis, N.; Moushi, Eleni E.; Tasiopoulos, Anastasios J.; Douvalis, A.; Papachristodoulou, C.; Hatzidimitriou, Antonios G.; Bakas, T.; Hadjikakou, Sotiris K. (Royal Society of Chemistry, 2020-09-07)
      The metalloantibiotic of formula Ph2Sn(CIP)2 (CIPTIN) (HCIP = ciprofloxacin) was synthesized by reacting ciprofloxacin hydrochloride (HCIP·HCl) (an antibiotic in clinical use) with diphenyltin dichloride (Ph2SnCl2DPTD). ...
    • Article  

      Drosophila melanogaster: A first step and a stepping-stone to anti-infectives 

      Tzelepis, Ilias; Kapsetaki, Stefania Elisavet; Panayidou, S.; Apidianakis, Yiorgos (2013)
      Following an expansion in the antibiotic drug discovery in the previous century, we now face a bottleneck in the production of new anti-infective drugs. Traditionally, chemical libraries are screened either using in vitro ...